GSK-137647A
更新时间:2023-02-25 12:44:31
采购接见:2次
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常用名 |
4-甲氧基-N-(2,4,6-三甲基苯)苯磺酰胺 |
CAS号 |
349085-82-1 |
价钱 |
¥需询单/1g ¥需询单/5g |
纯度 |
98.0% |
备货期 |
需询单 |
库存 |
现货 |
产物详情(用途,包装等) 用途: GSK137647A is a selective FFA4 agonist, with pEC50 of 6.3, 6.2, and 6.1 for human, Mouse and Rat FFA4, respectively.IC50 value: 6.3/6.2/6.1 (pEC50, for human/mouse/rat FFA4)Target: FFA4The pEC50s for Human , Mouse and Rat FFA1/2/3 are < 4.5. GSK137647A is evaluated against a panel of 65 targets in both full curve functional and binding assays and was shown to provide at least 100-fold selectivity against the panel which included 41 G-protein-coupled receptors (GPCRs), including additional members of the free fatty acid receptors (FFA1, FFA2, and FFA3). GSK137647A produces a concentration-dependent increase in glucose stimulated insulin secretion under high glucose conditions (25 mM). 物理化学性子: CAS号:349085-82-1 常用中文名:4-甲氧基-N-(2,4,6-三甲基苯)苯磺酰胺 常用英文名:GSK137647A 分子式:C16H19NO3S 分子量:305.39200 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A |
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