PF-05089771
更新时间:2022-08-21 16:09:40
采购接见:1次
|
常用名 |
PF-05089771 |
CAS号 |
1430806-04-4 |
价钱 |
¥需询单/10mg ¥需询单/1g |
纯度 |
98.9% |
备货期 |
需询单 |
库存 |
询单 |
产物详情(用途,包装等) 用途: PF-05089771 is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 11 nM, >1,000-fold selectivity over Nav1.3, 1.4 and Nav1.5, 1.8; interacts with the voltage-sensor domain (VSD) of domain IV, blocks all Nav1.7 splice variants with similar potency (5N11L, 5A11S, 5A11L and 5N11S, IC50s=11=33 nM); displays high selectivity over L-type calcium channels, KvLQT and hERG potassium channels; demonstrates in vivo efficacy in a mouse capsaicin-induced neurogenic flare model. Pain Phase 1 Discontinued 物理化学性子: CAS号:1430806-04-4 常用中文名:PF-05089771 常用英文名:PF 05089771 分子式:C18H12Cl2FN5O3S2 分子量:672.556 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A |
|