Raloxifene 6-glucuronide
更新时间:2020-12-18 22:54:27
采购访问:1次
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常用名 |
雷洛昔芬-6-葡萄糖醛酸苷 |
CAS号 |
174264-50-7 |
价格 |
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纯度 |
98.0% |
备货期 |
3天 |
库存 |
现货 |
产品网页 |
http://www.dcchemicals.com/product_show-Raloxifene-6-glucuronide.html |
产品详情(用途,包装等) Raloxifene 6-glucuronide is a primary metabolite of Raloxifene. Raloxifene 6-glucuronide is mediated mostly by UGT1A1 and UGT1A8. Raloxifene 6-glucuronide binds to estrogen receptor with an IC50 of 290 μM. Raloxifene is a selective and nonsteroidal estrogen receptor modulator. Raloxifene activates TGFβ3 promoter as a full agonist at nanomolar concentrations, and inhibits the estrogen response element-containing vitellogenin promoter expression. |
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