SKF-83566
更新时间:2020-12-18 22:54:27
采购访问:1次
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常用名 |
8-溴-2,3,4,5-四氢-3-甲基-5-苯基-1H-3-苯并氮杂-7-醇 |
CAS号 |
99295-33-7 |
价格 |
$需询单/250mg $需询单/100mg $需询单/1g |
纯度 |
98.0% |
备货期 |
3天 |
库存 |
现货 |
产品网页 |
http://www.dcchemicals.com/product_show-SKF-83566.html |
产品详情(用途,包装等) SKF-83566 is a potent,?blood-brain permeable and orally active D1-like dopamine receptor (D1DR)?antagonist and a weaker competitive antagonist at the vascular 5-HT2?receptor (Ki=11 nM). SKF-83566 is a competitive DAT (dopamine transporter) inhibitor with an IC50?of 5.7 μM. SKF-83566 also shows selective inhibition for adenylyl cyclase 2 (AC2) over AC1 and AC5 in the isolated rabbit thoracic aorta. SKF-83566 can be used for research of parkinson’s disease and nicotine craving alleviation. |
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