COL-144 (Lasmiditan) succinate
更新时间:2020-12-18 22:54:27
采购访问:1次
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常用名 |
Lasmiditan hemisuccinate |
CAS号 |
439239-92-6 |
价格 |
$500.0/100mg $900.0/250mg $1800.0/1g |
纯度 |
98.0% |
备货期 |
3天 |
库存 |
现货 |
产品网页 |
http://www.dcchemicals.com/product_show-COL-144_succinate.html |
产品详情(用途,包装等) Lasmiditan, also known as COL-144 and LY573144, is a novel, centrally acting, highly selective 5-HT(1F) receptor agonist (K1=2.21 μM) without vasoconstrictor activity that seemed effective when given as an intravenous infusion in a proof-of-concept migraine study. Lasmiditan showed efficacy in its primary endpoint, with a 2-hour placebo-subtracted headache response of 28.8%, though with frequent reports of dizziness, paresthesias, and vertigo. |
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